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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T62018 | Adenosine receptor inhibitor 2 | ||
Adenosine receptor inhibitor 2 (compound 14b) is a potent inhibitor of AR (adenosine receptor). Adenosine receptor inhibitor 2 exhibits dual affinity toward A 1 /A 2A ARs with higher affinity for the A 1 - than the A 2A ... | |||
T12163 | N6-(2-Phenylethyl)adenosine | N6-Phenethyladenosine,N6-Phenylethyladenosine | Adenosine Receptor |
N6-(2-Phenylethyl)adenosine (N6-Phenethyladenosine) is an adenosine derivative and an agonist of adenosine receptors with Ki values of 11.8 nM and 30.1 nM for rat and human A1. | |||
T5940 | Proxyphylline | 7-(2-Hydroxypropyl)theophylline | PDE , Adenosine Receptor |
Proxyphylline (7-(2-Hydroxypropyl)theophylline) is a dual of adenosine A1/A2a receptor inhibitor and phosphodiesterase (PDE) inhibitor. Proxyphylline acts as a cardiac stimulant, vasodilator and bronchodilator. | |||
T6884 | Namodenoson | 2-Cl-IB-MECA,CF-102 | Adenosine Receptor |
Namodenoson (2-Cl-IB-MECA) is an adenosine A3 receptor agonist. | |||
T23336 | SCH442416 | SCH 442416 | Adenosine Receptor |
SCH442416 (SCH 442416) is an selective antagonist of adenosine A2A receptor. SCH442416 binds to human and rat A2A receptors with high affinity (Ki values are 0.048 and 0.5 nM respectively). | |||
T9330 | MIPS521 | {2-Amino-4-[3,5-bis(trifluoromethyl)phenyl]thiophen-3-yl}(4-chlorophenyl)methanone | Adenosine Receptor |
MIPS521 ({2-Amino-4-[3,5-bis(trifluoromethyl)phenyl]thiophen-3-yl}(4-chlorophenyl)methanone) is a positive allosteric modulator of the A1R. | |||
T9516 | Binodenoson | WRC 0470,MRE-0470,2-(cyclohexylmethylidenehydrazino)adenos | Adenosine Receptor |
Binodenoson (WRC 0470) is a potent and selective A2A adenosine receptor agonist (KD=270 nM). Binodenoson is being developed as a short-acting coronary vasodilator as an adjunct to radiotracers for use in myocardial stres... | |||
T7320 | Tozadenant | SYN115 | Adenosine Receptor |
Tozadenant (SYN115) is an adenosine A2A receptor antagonist(Ki of 11.5 nM and 6 nM on human and rhesus,respectively) | |||
T29112 | VPC171 | VPC 171,VPC-171 | Adenosine Receptor |
VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM). | |||
T37793 | A2B receptor antagonist 2 | A2B receptor antagonist 2 | Adenosine Receptor |
A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B). | |||
T34685 | Sonedenoson | MRE 0094,MRE0094,MRE-0094 | SARS-CoV , Adenosine Receptor |
Sonedenoson (MRE0094) is an adenosine A(2A) receptor agonist and potential inhibitor potentially targeting SARS-CoV-2 coronavirus 2;-O-ribose methyltransferase, and may be used in the study of diabetic foot ulcers. | |||
T35573 | Adenosine 5’-methylenediphosphate (hydrate) | ||
Adenosine 5’-methylenediphosphate is an inhibitor of ecto-5’-nucleotidase, also known as CD73, with a Kivalue of 37 nM.1It inhibits cAMP accumulation induced by adenosine 5’-monophosphate , adenosine 5’-diphosphate , or ... | |||
T60511 | Theophylline sodium glycinate | ||
Theophylline (1,3-Dimethylxanthine) sodium glycinate is a potent inhibitor of phosphodiesterase (PDE) that inhibits PDE3 activity to relax airway smooth muscle. Theophylline sodium glycinate can be used for the research ... |