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Search Results for " adenosine receptor inhibitor 2 "

13

Compounds

Cat No. Product Name Synonyms Targets
T62018 Adenosine receptor inhibitor 2
Adenosine receptor inhibitor 2 (compound 14b) is a potent inhibitor of AR (adenosine receptor). Adenosine receptor inhibitor 2 exhibits dual affinity toward A 1 /A 2A ARs with higher affinity for the A 1 - than the A 2A ...
T12163 N6-(2-Phenylethyl)adenosine N6-Phenethyladenosine,N6-Phenylethyladenosine Adenosine Receptor
N6-(2-Phenylethyl)adenosine (N6-Phenethyladenosine) is an adenosine derivative and an agonist of adenosine receptors with Ki values of 11.8 nM and 30.1 nM for rat and human A1.
T5940 Proxyphylline 7-(2-Hydroxypropyl)theophylline PDE , Adenosine Receptor
Proxyphylline (7-(2-Hydroxypropyl)theophylline) is a dual of adenosine A1/A2a receptor inhibitor and phosphodiesterase (PDE) inhibitor. Proxyphylline acts as a cardiac stimulant, vasodilator and bronchodilator.
T6884 Namodenoson 2-Cl-IB-MECA,CF-102 Adenosine Receptor
Namodenoson (2-Cl-IB-MECA) is an adenosine A3 receptor agonist.
T23336 SCH442416 SCH 442416 Adenosine Receptor
SCH442416 (SCH 442416) is an selective antagonist of adenosine A2A receptor. SCH442416 binds to human and rat A2A receptors with high affinity (Ki values are 0.048 and 0.5 nM respectively).
T9330 MIPS521 {2-Amino-4-[3,5-bis(trifluoromethyl)phenyl]thiophen-3-yl}(4-chlorophenyl)methanone Adenosine Receptor
MIPS521 ({2-Amino-4-[3,5-bis(trifluoromethyl)phenyl]thiophen-3-yl}(4-chlorophenyl)methanone) is a positive allosteric modulator of the A1R.
T9516 Binodenoson WRC 0470,MRE-0470,2-(cyclohexylmethylidenehydrazino)adenos Adenosine Receptor
Binodenoson (WRC 0470) is a potent and selective A2A adenosine receptor agonist (KD=270 nM). Binodenoson is being developed as a short-acting coronary vasodilator as an adjunct to radiotracers for use in myocardial stres...
T7320 Tozadenant SYN115 Adenosine Receptor
Tozadenant (SYN115) is an adenosine A2A receptor antagonist(Ki of 11.5 nM and 6 nM on human and rhesus,respectively)
T29112 VPC171 VPC 171,VPC-171 Adenosine Receptor
VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).
T37793 A2B receptor antagonist 2 A2B receptor antagonist 2 Adenosine Receptor
A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).
T34685 Sonedenoson MRE 0094,MRE0094,MRE-0094 SARS-CoV , Adenosine Receptor
Sonedenoson (MRE0094) is an adenosine A(2A) receptor agonist and potential inhibitor potentially targeting SARS-CoV-2 coronavirus 2;-O-ribose methyltransferase, and may be used in the study of diabetic foot ulcers.
T35573 Adenosine 5’-methylenediphosphate (hydrate)
Adenosine 5’-methylenediphosphate is an inhibitor of ecto-5’-nucleotidase, also known as CD73, with a Kivalue of 37 nM.1It inhibits cAMP accumulation induced by adenosine 5’-monophosphate , adenosine 5’-diphosphate , or ...
T60511 Theophylline sodium glycinate
Theophylline (1,3-Dimethylxanthine) sodium glycinate is a potent inhibitor of phosphodiesterase (PDE) that inhibits PDE3 activity to relax airway smooth muscle. Theophylline sodium glycinate can be used for the research ...
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